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Bay 59-3074
CAS No. 406205-74-1
Bay 59-3074 ( Bay59-3074;Bay-59-3074 )
Catalog No. M14399 CAS No. 406205-74-1
A potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 35 | In Stock |
|
| 10MG | 58 | In Stock |
|
| 25MG | 110 | In Stock |
|
| 50MG | 178 | In Stock |
|
| 100MG | 332 | In Stock |
|
| 200MG | 494 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBay 59-3074
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively.
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DescriptionA potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively; displays antihyperalgesic and antiallodynic effects against thermal or mechanical stimuli in rat models of chronic neuropathic; orally acitve.
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SynonymsBay59-3074;Bay-59-3074
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCB1;CB2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number406205-74-1
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Formula Weight453.36
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Molecular FormulaC18H13F6NO4S
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 34 mg/mL
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SMILESO=S(CCCC(F)(F)F)(OC1=CC=CC(OC2=CC=CC(C(F)(F)F)=C2C#N)=C1)=O
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Chemical Name1-Butanesulfonic acid, 4,4,4-trifluoro-, 3-[2-cyano-3-(trifluoromethyl)phenoxy]phenyl ester
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. De Vry J, et al. J Pharmacol Exp Ther. 2004 Aug;310(2):620-32.
2. De Vry J, et al. Eur J Pharmacol. 2004 Nov 28;505(1-3):127-33.
3. Teng H, et al. Bioorg Med Chem Lett. 2011 Oct 1;21(19):5999-6002.
2. De Vry J, et al. Eur J Pharmacol. 2004 Nov 28;505(1-3):127-33.
3. Teng H, et al. Bioorg Med Chem Lett. 2011 Oct 1;21(19):5999-6002.
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Bay 59-3074
A potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively.
